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PDB: 1 results

5VDK
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BU of 5vdk by Molmil
Crystal structure of human WEE2 kinase domain in complex with MK1775
Descriptor: 1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3H-pyrazolo[3,4-d]pyrimidin-3-one, PHOSPHATE ION, Wee1-like protein kinase 2
Authors:Zhu, J.-Y, Schonbrunn, E.
Deposit date:2017-04-03
Release date:2017-08-23
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Structural Basis of Wee Kinases Functionality and Inactivation by Diverse Small Molecule Inhibitors.
J. Med. Chem., 60, 2017

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