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PDB: 1 results

Human alpha-thrombin complexed with N-(methylsulfonyl)-D-phenylalanyl-N-((1-carbamimidoyl-4-piperidinyl)methyl)-l-prolinamide (BMS-189664)
Descriptor:	Hirudin variant-2, N-(methylsulfonyl)-D-phenylalanyl-N-[(1-carbamimidoylpiperidin-4-yl)methyl]-L-prolinamide, Prothrombin
Authors:	Malley, M, Sack, J.S.
Deposit date:	2011-09-16
Release date:	2011-10-12
Last modified:	2012-12-12
Method:	X-RAY DIFFRACTION (2.49 Å)
Cite:	Molecular design and structure-activity relationships leading to the potent, selective, and orally active thrombin active site inhibitor BMS-189664. Bioorg.Med.Chem.Lett., 12, 2002