8OO8
 
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9FLF
 | | Three-Dimensional Structure of Human Carbonic Anhydrase IX in Complex with a Covalent Inhibitor | | Descriptor: | 3-[[(1~{R},4~{Z})-cyclododec-4-en-1-yl]amino]-4-ethylsulfonyl-2,5,6-tris(fluoranyl)benzenesulfonamide, Carbonic anhydrase, ZINC ION | | Authors: | Leitans, J, Tars, K. | | Deposit date: | 2024-06-05 | | Release date: | 2024-12-18 | | Last modified: | 2025-01-22 | | Method: | X-RAY DIFFRACTION (2.2 Å) | | Cite: | Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX.
Elife, 13, 2024
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8S4F
 | | Human carbonic anhydrase I covalently bound to AV21-08 | | Descriptor: | 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 3-(cyclooctylamino)-4-ethylsulfonyl-2,5,6-tris(fluoranyl)benzenesulfonamide, ... | | Authors: | Manakova, E.N, Grazulis, S, Paketuryte-Latve, V, Vaskevicius, A, Smirnov, A. | | Deposit date: | 2024-02-21 | | Release date: | 2024-12-18 | | Last modified: | 2025-01-22 | | Method: | X-RAY DIFFRACTION (1.39 Å) | | Cite: | Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX.
Elife, 13, 2024
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