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PDB: 1 results

HIV-1 Integrase catalytic core domain complexed with allosteric inhibitor STP03-0404
Descriptor:	(2S)-tert-butoxy{4-(4-chlorophenyl)-2,3,6-trimethyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-5-yl}acetic acid, Integrase
Authors:	Lindenberger, J.J, Kvaratskhelia, M.
Deposit date:	2020-10-09
Release date:	2021-09-22
Last modified:	2023-10-18
Method:	X-RAY DIFFRACTION (2.19 Å)
Cite:	A highly potent and safe pyrrolopyridine-based allosteric HIV-1 integrase inhibitor targeting host LEDGF/p75-integrase interaction site. Plos Pathog., 17, 2021