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PDB: 2 results

8FLN
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BU of 8fln by Molmil
Crystal structure of BTK C481S kinase domain in complex with pirtobrutinib
Descriptor: 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, GLYCEROL, SULFATE ION, ...
Authors:Cedervall, E.P, Morales, T.H, Allerston, C.K.
Deposit date:2022-12-21
Release date:2023-03-01
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (1.334 Å)
Cite:Preclinical characterization of pirtobrutinib, a highly selective, noncovalent (reversible) BTK inhibitor.
Blood, 142, 2023
8FLL
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BU of 8fll by Molmil
Crystal structure of BTK kinase domain in complex with pirtobrutinib
Descriptor: 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, GLYCEROL, SULFATE ION, ...
Authors:Cedervall, E.P, Morales, T.H, Allerston, C.K.
Deposit date:2022-12-21
Release date:2023-03-01
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.498 Å)
Cite:Preclinical characterization of pirtobrutinib, a highly selective, noncovalent (reversible) BTK inhibitor.
Blood, 142, 2023

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PDB entries from 2024-07-17

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