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PDB: 1 results
8STG
Discovery and clinical validation of RLY-4008, the first highly selective FGFR2 inhibitor with activity across FGFR2 alterations and resistance mutations
Descriptor:
Fibroblast growth factor receptor 2, N-{4-[(5P)-4-amino-5-{3-fluoro-4-[(4-methylpyrimidin-2-yl)oxy]phenyl}-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}-2-methylpropanamide
Authors:
Valverde, R
,
Foster, L.
Deposit date:
2023-05-10
Release date:
2023-06-07
Last modified:
2023-10-25
Method:
X-RAY DIFFRACTION (3.79 Å)
Cite:
RLY-4008, the First Highly Selective FGFR2 Inhibitor with Activity across FGFR2 Alterations and Resistance Mutations.
Cancer Discov, 13, 2023
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PDB entries from 2024-07-03