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PDB: 1 results

8E4A
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BU of 8e4a by Molmil
Pseudomonas LpxC in complex with LPC-233
Descriptor: 4-(4-cyclopropylbuta-1,3-diyn-1-yl)-N-[(2S,3S)-4,4-difluoro-3-hydroxy-1-(hydroxyamino)-3-methyl-1-oxobutan-2-yl]benzamide, UDP-3-O-acyl-N-acetylglucosamine deacetylase, ZINC ION
Authors:Najeeb, J, Zhou, P.
Deposit date:2022-08-17
Release date:2023-08-23
Method:X-RAY DIFFRACTION (2.034 Å)
Cite:Preclinical safety and efficacy characterization of an LpxC inhibitor against Gram-negative pathogens.
Sci Transl Med, 15, 2023

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