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PDB: 3 件

3MJ2
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BU of 3mj2 by Molmil
X-ray crystal structure of ITK complexed with inhibitor BMS-509744
分子名称: N-[5-({5-[(4-acetylpiperazin-1-yl)carbonyl]-4-methoxy-2-methylphenyl}sulfanyl)-1,3-thiazol-2-yl]-4-({[(1S)-1,2,2-trimethylpropyl]amino}methyl)benzamide, Tyrosine-protein kinase ITK/TSK
著者Kuglstatter, A, Villasenor, A.G.
登録日2010-04-12
公開日2010-06-30
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structures of IL-2-inducible T cell kinase complexed with inhibitors: insights into rational drug design and activity regulation.
Chem.Biol.Drug Des., 76, 2010
3MJ1
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BU of 3mj1 by Molmil
X-ray crystal structure of ITK complexed with inhibitor RO5191614
分子名称: 7-[(4-methylpiperazin-1-yl)methyl]-4-[(3-methyl-1H-pyrazol-5-yl)amino]-2-(tetrahydro-2H-pyran-4-yl)phthalazin-1(2H)-one, Tyrosine-protein kinase ITK/TSK
著者Kuglstatter, A, Villasenor, A.G.
登録日2010-04-12
公開日2010-06-30
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献Crystal structures of IL-2-inducible T cell kinase complexed with inhibitors: insights into rational drug design and activity regulation.
Chem.Biol.Drug Des., 76, 2010
3MIY
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BU of 3miy by Molmil
X-ray crystal structure of ITK complexed with sunitinib
分子名称: N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carbo xamide, Tyrosine-protein kinase ITK/TSK
著者Kuglstatter, A, Villasenor, A.G.
登録日2010-04-12
公開日2010-06-30
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献Crystal structures of IL-2-inducible T cell kinase complexed with inhibitors: insights into rational drug design and activity regulation.
Chem.Biol.Drug Des., 76, 2010

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件を2024-05-15に公開中

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