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PDB: 2 results
8OOD
Crystal structure of human DCAF1 WD40 repeats (Q1250L) in complex with compound 15
Descriptor:
1,2-ETHANEDIOL, ACETATE ION, DDB1- and CUL4-associated factor 1, ...
Authors:
Schroeder, M
,
Renatus, M.
Deposit date:
2023-04-05
Release date:
2023-05-24
Last modified:
2024-06-19
Method:
X-RAY DIFFRACTION (1.497 Å)
Cite:
Reinstating targeted protein degradation with DCAF1 PROTACs in CRBN PROTAC resistant settings
Biorxiv, 2023
8OO5
Crystal structure of human DCAF1 WD40 repeats (Q1250L) in complex with compound 13
Descriptor:
1,2-ETHANEDIOL, 1-[4-[4-(2-azanylethylamino)-2-[1-(4-chlorophenyl)cyclohexyl]quinazolin-7-yl]piperazin-1-yl]ethanone, DDB1- and CUL4-associated factor 1
Authors:
Schroeder, M
,
Renatus, M.
Deposit date:
2023-04-04
Release date:
2023-05-24
Last modified:
2024-06-19
Method:
X-RAY DIFFRACTION (2.25 Å)
Cite:
Reinstating targeted protein degradation with DCAF1 PROTACs in CRBN PROTAC resistant settings
Biorxiv, 2023
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222415
PDB entries from 2024-07-10