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PDB: 1 results

4KCG
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BU of 4kcg by Molmil
Human dCK C4S-S74E mutant in complex with UDP and the DI-39 inhibitor
Descriptor: Deoxycytidine kinase, N-{2-[5-(4-{[(4,6-diaminopyrimidin-2-yl)sulfanyl]methyl}-5-propyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]ethyl}methanesulfonamide, URIDINE-5'-DIPHOSPHATE
Authors:Nomme, J, Lavie, A.
Deposit date:2013-04-24
Release date:2014-03-12
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2.09 Å)
Cite:Co-targeting of convergent nucleotide biosynthetic pathways for leukemia eradication.
J.Exp.Med., 211, 2014

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