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PDB: 3 件

6M11
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BU of 6m11 by Molmil
Crystal structure of Rnase L in complex with Sunitinib
分子名称: 5'-O-MONOPHOSPHORYLADENYLYL(2'->5')ADENYLYL(2'->5')ADENOSINE, N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carbo xamide, PHOSPHATE ION, ...
著者Tang, J, Huang, H.
登録日2020-02-24
公開日2020-09-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.46 Å)
主引用文献Sunitinib inhibits RNase L by destabilizing its active dimer conformation.
Biochem.J., 477, 2020
6M12
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BU of 6m12 by Molmil
Crystal Structure of Rnase L in complex with SU11652
分子名称: 5-[(E)-(5-CHLORO-2-OXO-1,2-DIHYDRO-3H-INDOL-3-YLIDENE)METHYL]-N-[2-(DIETHYLAMINO)ETHYL]-2,4-DIMETHYL-1H-PYRROLE-3-CARBOXAMIDE, PHOSPHATE ION, Ribonuclease L, ...
著者Tang, J, Huang, H.
登録日2020-02-24
公開日2020-09-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Sunitinib inhibits RNase L by destabilizing its active dimer conformation.
Biochem.J., 477, 2020
6M13
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BU of 6m13 by Molmil
Crystal structure of Rnase L in complex with Toceranib
分子名称: 5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-ylidene)methyl]-2,4-dimethyl-N-(2-pyrrolidin-1-ylethyl)-1H-pyrrole-3-carboxamide, PHOSPHATE ION, Ribonuclease L, ...
著者Tang, J, Huang, H.
登録日2020-02-24
公開日2020-09-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.56 Å)
主引用文献Sunitinib inhibits RNase L by destabilizing its active dimer conformation.
Biochem.J., 477, 2020

220113

件を2024-05-22に公開中

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