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PDB: 1 results

8A92
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BU of 8a92 by Molmil
p53-Y220C Core Domain in Complex with a Bromo-trifluoro-pyrazole-amine
Descriptor: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 4-bromanyl-5-(trifluoromethyl)-1H-pyrazol-3-amine, Cellular tumor antigen p53, ...
Authors:Stahlecker, J, Braun, M.B, Stehle, T, Boeckler, F.M.
Deposit date:2022-06-27
Release date:2022-11-09
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.37 Å)
Cite:Revisiting a challenging p53 binding site: a diversity-optimized HEFLib reveals diverse binding modes in T-p53C-Y220C.
Rsc Med Chem, 13, 2022

221716

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