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PDB: 1 results
7FIC
Reversible lysine-targeted probes reveal residence time-based kinase selectivity in vivo
Descriptor:
6-[(5-cyclopropyl-1~{H}-pyrazol-3-yl)amino]-2-[4-[(3-methyl-4-oxidanyl-phenyl)methyl]piperazin-1-yl]-~{N}-prop-2-ynyl-pyrimidine-4-carboxamide, Aurora kinase A, CHLORIDE ION
Authors:
Craven, G.B
,
Wan, X.B
,
Taunton, J.
Deposit date:
2021-07-31
Release date:
2022-06-08
Last modified:
2023-11-29
Method:
X-RAY DIFFRACTION (2.32 Å)
Cite:
Reversible lysine-targeted probes reveal residence time-based kinase selectivity.
Nat.Chem.Biol., 18, 2022
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PDB entries from 2024-07-10