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PDB: 4 results

9CT4
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BU of 9ct4 by Molmil
HsSTING with diABZI and C53, curved conformation
Descriptor: 1-[(2-chloro-6-fluorophenyl)methyl]-3,3-dimethyl-2-oxo-N-[(2,4,6-trifluorophenyl)methyl]-2,3-dihydro-1H-indole-6-carboxamide, 1-[(2E)-4-{5-carbamoyl-2-[(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)amino]-7-methoxy-1H-1,3-benzimidazol-1-yl}but-2-en-1-yl]-2-[(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)amino]-7-[3-(morpholin-4-yl)propoxy]-1H-1,3-benzimidazole-5-carboxamide, Stimulator of interferon genes protein
Authors:Gharpure, A, Sulpizio, A, Lairson, L.L, Ward, A.B.
Deposit date:2024-07-24
Release date:2025-04-23
Method:ELECTRON MICROSCOPY (3.29 Å)
Cite:Distinct oligomeric assemblies of STING induced by non-nucleotide agonists.
Nat Commun, 16, 2025
9CT3
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BU of 9ct3 by Molmil
HsSTING with SR-717 and C53
Descriptor: 1-[(2-chloro-6-fluorophenyl)methyl]-3,3-dimethyl-2-oxo-N-[(2,4,6-trifluorophenyl)methyl]-2,3-dihydro-1H-indole-6-carboxamide, 4,5-difluoro-2-{[6-(1H-imidazol-1-yl)pyridazine-3-carbonyl]amino}benzoic acid, Stimulator of interferon genes protein
Authors:Gharpure, A, Sulpizio, A, Lairson, L.L, Ward, A.B.
Deposit date:2024-07-24
Release date:2025-04-23
Method:ELECTRON MICROSCOPY (3.09 Å)
Cite:Distinct oligomeric assemblies of STING induced by non-nucleotide agonists.
Nat Commun, 16, 2025
9CT6
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BU of 9ct6 by Molmil
HsSTING with diABZI and C53, apart conformation
Descriptor: 1-[(2-chloro-6-fluorophenyl)methyl]-3,3-dimethyl-2-oxo-N-[(2,4,6-trifluorophenyl)methyl]-2,3-dihydro-1H-indole-6-carboxamide, 1-[(2E)-4-{5-carbamoyl-2-[(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)amino]-7-methoxy-1H-1,3-benzimidazol-1-yl}but-2-en-1-yl]-2-[(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)amino]-7-[3-(morpholin-4-yl)propoxy]-1H-1,3-benzimidazole-5-carboxamide, Stimulator of interferon genes protein
Authors:Gharpure, A, Sulpizio, A, Lairson, L.L, Ward, A.B.
Deposit date:2024-07-24
Release date:2025-04-23
Method:ELECTRON MICROSCOPY (3.56 Å)
Cite:Distinct oligomeric assemblies of STING induced by non-nucleotide agonists.
Nat Commun, 16, 2025
9CT5
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BU of 9ct5 by Molmil
HsSTING with diABZI and C53, together conformation
Descriptor: 1-[(2-chloro-6-fluorophenyl)methyl]-3,3-dimethyl-2-oxo-N-[(2,4,6-trifluorophenyl)methyl]-2,3-dihydro-1H-indole-6-carboxamide, 1-[(2E)-4-{5-carbamoyl-2-[(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)amino]-7-methoxy-1H-1,3-benzimidazol-1-yl}but-2-en-1-yl]-2-[(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)amino]-7-[3-(morpholin-4-yl)propoxy]-1H-1,3-benzimidazole-5-carboxamide, Stimulator of interferon genes protein
Authors:Gharpure, A, Sulpizio, A, Lairson, L.L, Ward, A.B.
Deposit date:2024-07-24
Release date:2025-04-23
Method:ELECTRON MICROSCOPY (3.67 Å)
Cite:Distinct oligomeric assemblies of STING induced by non-nucleotide agonists.
Nat Commun, 16, 2025

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PDB entries from 2025-07-09

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