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PDB: 2 results
1YCI
Factor inhibiting HIF-1 alpha in complex with N-(carboxycarbonyl)-D-phenylalanine
Descriptor:
FE (II) ION, Hypoxia-inducible factor 1 alpha inhibitor, N-(CARBOXYCARBONYL)-D-PHENYLALANINE, ...
Authors:
McDonough, M.A
,
Schofield, C.J.
Deposit date:
2004-12-22
Release date:
2005-05-31
Last modified:
2023-10-25
Method:
X-RAY DIFFRACTION (2.7 Å)
Cite:
Selective inhibition of factor inhibiting hypoxia-inducible factor
J.Am.Chem.Soc., 127, 2005
2ILM
Factor Inhibiting HIF-1 Alpha D201A Mutant in Complex with FE(II), Alpha-Ketoglutarate and HIF-1 Alpha 35mer
Descriptor:
2-OXOGLUTARIC ACID, BICARBONATE ION, FE (II) ION, ...
Authors:
Mcdonough, M.A
,
Schofield, C.J.
Deposit date:
2006-10-03
Release date:
2007-08-14
Last modified:
2023-08-30
Method:
X-RAY DIFFRACTION (2.3 Å)
Cite:
Evidence that two enzyme-derived histidine ligands are sufficient for iron binding and catalysis by factor inhibiting HIF (FIH).
J.Biol.Chem., 283, 2008
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PDB entries from 2024-07-10