Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 1 results

6TCU
DownloadVisualize
BU of 6tcu by Molmil
Glycogen synthase kinase-3 beta (GSK3b) in complex with ligand 1
Descriptor: 5-[2,3-bis(fluoranyl)phenyl]-~{N}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{H}-indazole-3-carboxamide, ACETATE ION, Glycogen synthase kinase-3 beta
Authors:Lammens, A, Krapp, S, Buonfiglio, R, Ombrato, R.
Deposit date:2019-11-06
Release date:2020-09-16
Method:X-RAY DIFFRACTION (2.14 Å)
Cite:Optimization of Indazole-Based GSK-3 Inhibitors with Mitigated hERG Issue andIn VivoActivity in a Mood Disorder Model.
Acs Med.Chem.Lett., 11, 2020

222036

PDB entries from 2024-07-03

PDB statisticsPDBj update infoContact PDBjnumon