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PDB: 1 results

6ILZ
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BU of 6ilz by Molmil
Crystal structure of PKCiota in complex with inhibitor
Descriptor: 2-amino-5-[3-(piperazin-1-yl)phenyl]-N-(pyridin-4-yl)pyridine-3-carboxamide, Protein kinase C iota type
Authors:Baburajendran, N, Hill, J.
Deposit date:2018-10-21
Release date:2019-06-26
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (3.261 Å)
Cite:Fragment-based Discovery of a Small-Molecule Protein Kinase C-iota Inhibitor Binding Post-kinase Domain Residues.
Acs Med.Chem.Lett., 10, 2019

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