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PDB: 3 results

5UT6
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BU of 5ut6 by Molmil
JAK2 JH2 in complex with a diaminopyrimidine
Descriptor: 4-({4-amino-6-[3-(hydroxymethyl)-1H-pyrazol-1-yl]pyrimidin-2-yl}amino)benzonitrile, ACETATE ION, DIMETHYL SULFOXIDE, ...
Authors:Puleo, D.E, Schlessinger, J.
Deposit date:2017-02-14
Release date:2017-06-07
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.645 Å)
Cite:JAK2 JH2 Fluorescence Polarization Assay and Crystal Structures for Complexes with Three Small Molecules.
ACS Med Chem Lett, 8, 2017
5UT5
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BU of 5ut5 by Molmil
JAK2 JH2 in complex with GLPG0634
Descriptor: ACETATE ION, DIMETHYL SULFOXIDE, GLYCEROL, ...
Authors:Puleo, D.E, Schlessinger, J.
Deposit date:2017-02-14
Release date:2017-06-07
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:JAK2 JH2 Fluorescence Polarization Assay and Crystal Structures for Complexes with Three Small Molecules.
ACS Med Chem Lett, 8, 2017
5UT4
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BU of 5ut4 by Molmil
JAK2 JH2 in complex with NVP-BSK805
Descriptor: 8-[3,5-difluoro-4-(morpholin-4-ylmethyl)phenyl]-2-(1-piperidin-4-yl-1H-pyrazol-4-yl)quinoxaline, DIMETHYL SULFOXIDE, GLYCEROL, ...
Authors:Puleo, D.E, Schlessinger, J.
Deposit date:2017-02-14
Release date:2017-06-07
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2 Å)
Cite:JAK2 JH2 Fluorescence Polarization Assay and Crystal Structures for Complexes with Three Small Molecules.
ACS Med Chem Lett, 8, 2017

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