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PDB: 1 results

8EME
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BU of 8eme by Molmil
EGFR(T790M/V948R) in complex with ZNL-0056
Descriptor: Epidermal growth factor receptor, N-{7-methyl-1-[(3S)-1-(prop-2-enoyl)azepan-3-yl]-1H-benzimidazol-2-yl}-5-(prop-2-enamido)thiophene-3-carboxamide
Authors:Beyett, T.S, Eck, M.J.
Deposit date:2022-09-27
Release date:2023-10-18
Last modified:2024-07-10
Method:X-RAY DIFFRACTION (3.32 Å)
Cite:Molecular Bidents with Two Electrophilic Warheads as a New Pharmacological Modality.
Acs Cent.Sci., 10, 2024

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PDB entries from 2024-10-16

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