9DCD
 
 | | Structure of J-PKAc chimera in complex with Aplithianine d2 | | Descriptor: | N-(2-aminoethyl)-4-(7H-purin-6-yl)-3,4-dihydro-2H-1,4-thiazine-6-carboxamide, cAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase inhibitor alpha | | Authors: | Martinez Fiesco, J.A, Zhang, P. | | Deposit date: | 2024-08-25 | | Release date: | 2025-07-09 | | Method: | X-RAY DIFFRACTION (2.7 Å) | | Cite: | Chemical Evolution of Aplithianine Class of Serine/Threonine Kinase Inhibitors.
J.Med.Chem., 68, 2025
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9DC6
 | | Structure of J-PKAc chimera in complex with Aplithianine e1 | | Descriptor: | N-(2-aminoethyl)-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-3,4-dihydro-2H-1,4-thiazine-6-carboxamide, cAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase inhibitor alpha | | Authors: | Martinez Fiesco, J.A, Zhang, P. | | Deposit date: | 2024-08-25 | | Release date: | 2025-07-09 | | Method: | X-RAY DIFFRACTION (2.7 Å) | | Cite: | Chemical Evolution of Aplithianine Class of Serine/Threonine Kinase Inhibitors.
J.Med.Chem., 68, 2025
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