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PDB: 1 results

7RA5
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BU of 7ra5 by Molmil
CDK2 IN COMPLEX WITH COMPOUND 4
Descriptor: 4-[7-(methanesulfonyl)-1H-indol-3-yl]-N-[(3S)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amine, Cyclin-dependent kinase 2
Authors:Marineau, J.J, Malojcic, G.
Deposit date:2021-06-30
Release date:2021-11-03
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (1.67 Å)
Cite:Discovery of SY-5609: A Selective, Noncovalent Inhibitor of CDK7.
J.Med.Chem., 65, 2022

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PDB entries from 2024-07-10

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