PDB Search results for query - Protein Data Bank Japan

PDB: 2 results

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 (3R,4R)-N-cyclohexyl-4-((3-methyl-2-oxo-1,2-dihydro-1,7-naphthyridin-8-yl)amino)piperidine-3-carboxamide
Descriptor:	(3R,4R)-N-cyclohexyl-4-((3-methyl-2-oxo-1,2-dihydro-1,7-naphthyridin-8-yl)amino)piperidine-3-carboxamide, Bromodomain-containing protein 4
Authors:	Chung, C.
Deposit date:	2020-05-31
Release date:	2020-07-29
Last modified:	2024-05-01
Method:	X-RAY DIFFRACTION (1.26 Å)
Cite:	GSK789: A Selective Inhibitor of the First Bromodomains (BD1) of the Bromo and Extra Terminal Domain (BET) Proteins. J.Med.Chem., 63, 2020

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 with GSK789
Descriptor:	(3~{R},4~{R})-~{N}-cyclohexyl-4-[[5-(furan-2-yl)-3-methyl-2-oxidanylidene-1~{H}-1,7-naphthyridin-8-yl]amino]-1-methyl-piperidine-3-carboxamide, Bromodomain-containing protein 4
Authors:	Chung, C.
Deposit date:	2020-05-31
Release date:	2020-07-29
Last modified:	2024-05-01
Method:	X-RAY DIFFRACTION (1.624 Å)
Cite:	GSK789: A Selective Inhibitor of the First Bromodomains (BD1) of the Bromo and Extra Terminal Domain (BET) Proteins. J.Med.Chem., 63, 2020