9QB5
 
 | | AP2-associated protein kinase 1 (AAK1) bound to CKJB68 | | Descriptor: | AP2-associated protein kinase 1, SULFATE ION, ~{N}-(phenylmethyl)-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamide | | Authors: | Preuss, F, Mensing, T.E, Hanke, T, Knapp, S, Mathea, S. | | Deposit date: | 2025-02-28 | | Release date: | 2025-04-09 | | Last modified: | 2025-10-22 | | Method: | X-RAY DIFFRACTION (2 Å) | | Cite: | Development of pyrazolo[1,5-a]pyrimidine based macrocyclic kinase inhibitors targeting AAK1.
Eur.J.Med.Chem., 299, 2025
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