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PDB: 1 results

6EK3
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BU of 6ek3 by Molmil
PARP15 CATALYTIC DOMAIN MUTANT (Y598L) IN COMPLEX WITH OUL35
Descriptor: 4-(4-aminocarbonylphenoxy)benzamide, Poly [ADP-ribose] polymerase 15
Authors:Maksimainen, M.M, Lehtio, L.
Deposit date:2017-09-25
Release date:2018-07-25
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:4-(Phenoxy) and 4-(benzyloxy)benzamides as potent and selective inhibitors of mono-ADP-ribosyltransferase PARP10/ARTD10.
Eur J Med Chem, 156, 2018

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