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PDB: 2 results

6BT5
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BU of 6bt5 by Molmil
Human mGlu8 Receptor complexed with L-AP4
Descriptor: (2S)-2-amino-4-phosphonobutanoic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, Metabotropic glutamate receptor 8
Authors:Schkeryantz, J.M, Chen, Q, Ho, J.D, Atwell, S, Zhang, A, Vargas, M.C, Wang, J, Monn, J.A, Hao, J.
Deposit date:2017-12-05
Release date:2018-02-07
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.92 Å)
Cite:Determination of L-AP4-bound human mGlu8 receptor amino terminal domain structure and the molecular basis for L-AP4's group III mGlu receptor functional potency and selectivity.
Bioorg. Med. Chem. Lett., 28, 2018
6BSZ
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BU of 6bsz by Molmil
Human mGlu8 Receptor complexed with glutamate
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, GLUTAMIC ACID, Metabotropic glutamate receptor 8, ...
Authors:Schkeryantz, J.M, Chen, Q, Ho, J.D, Atwell, S, Zhang, A, Vargas, M.C, Wang, J, Monn, J.A, Hao, J.
Deposit date:2017-12-04
Release date:2018-02-07
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.65 Å)
Cite:Determination of L-AP4-bound human mGlu8 receptor amino terminal domain structure and the molecular basis for L-AP4's group III mGlu receptor functional potency and selectivity.
Bioorg. Med. Chem. Lett., 28, 2018

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