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PDB: 4 results
5MQG
Crystal structure of CREBBP bromodomain complexed with CBP015
Descriptor:
1-(4-azanyl-3-methoxy-phenyl)ethanone, CREB-binding protein
Authors:
Zhu, J
,
Spiliotopoulos, D
,
Caflisch, A.
Deposit date:
2016-12-20
Release date:
2017-04-19
Last modified:
2024-05-08
Method:
X-RAY DIFFRACTION (1.35 Å)
Cite:
Virtual screen to NMR (VS2NMR): Discovery of fragment hits for the CBP bromodomain.
Bioorg. Med. Chem. Lett., 27, 2017
5MPZ
Crystal structure of CREBBP bromodomain complexed with CBP007
Descriptor:
CREB-binding protein, methyl 2-oxidanylidene-3~{H}-1,3-benzoxazole-6-carboxylate
Authors:
Zhu, J
,
Spiliotopoulos, D
,
Caflisch, A.
Deposit date:
2016-12-19
Release date:
2017-05-10
Last modified:
2024-05-08
Method:
X-RAY DIFFRACTION (1.4 Å)
Cite:
Virtual screen to NMR (VS2NMR): Discovery of fragment hits for the CBP bromodomain.
Bioorg. Med. Chem. Lett., 27, 2017
5MQE
Crystal structure of CREBBP bromodomain complexed with CBP006
Descriptor:
4-bromanyl-~{N}-methyl-1~{H}-pyrrole-2-carboxamide, CREB-binding protein
Authors:
Zhu, J
,
Spiliotopoulos, D
,
Caflisch, A.
Deposit date:
2016-12-20
Release date:
2017-04-19
Last modified:
2024-05-08
Method:
X-RAY DIFFRACTION (1.65 Å)
Cite:
Virtual screen to NMR (VS2NMR): Discovery of fragment hits for the CBP bromodomain.
Bioorg. Med. Chem. Lett., 27, 2017
5MQK
Crystal structure of CREBBP bromodomain complexed with CBP019
Descriptor:
1-(1-methylindol-3-yl)ethanone, CREB-binding protein
Authors:
Zhu, J
,
Spiliotopoulos, D
,
Caflisch, A.
Deposit date:
2016-12-20
Release date:
2017-04-19
Last modified:
2024-05-08
Method:
X-RAY DIFFRACTION (1.53 Å)
Cite:
Virtual screen to NMR (VS2NMR): Discovery of fragment hits for the CBP bromodomain.
Bioorg. Med. Chem. Lett., 27, 2017
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222926
PDB entries from 2024-07-24