PDB Search results for query - Protein Data Bank Japan

PDB: 2 results

Structure-based optimization of 1H-imidazole-2-carboxamides as Axl kinase inhibitors utilizing a Mer mutant surrogate
Descriptor:	N-(2-{4-[(2S)-4-(methylsulfonyl)morpholin-2-yl]-1,3-thiazol-2-yl}phenyl)-1H-imidazole-2-carboxamide, Tyrosine-protein kinase Mer
Authors:	Hoffman, I.D, Lawson, J.D.
Deposit date:	2016-09-13
Release date:	2017-01-25
Last modified:	2024-03-06
Method:	X-RAY DIFFRACTION (2.24 Å)
Cite:	Structure-based optimization of 1H-imidazole-2-carboxamides as Axl kinase inhibitors utilizing a Mer mutant surrogate. Bioorg. Med. Chem. Lett., 27, 2017

Structure-based optimization of 1H-imidazole-2-carboxamides as Axl kinase inhibitors utilizing a Mer mutant surrogate
Descriptor:	N-[2-{4-[(2S)-4-(methylsulfonyl)morpholin-2-yl]-1,3-thiazol-2-yl}-4-(morpholin-4-yl)phenyl]-1H-imidazole-2-carboxamide, Tyrosine-protein kinase Mer
Authors:	Hoffman, I.D, Lawson, J.D.
Deposit date:	2016-09-16
Release date:	2017-01-25
Last modified:	2024-03-06
Method:	X-RAY DIFFRACTION (2.68 Å)
Cite:	Structure-based optimization of 1H-imidazole-2-carboxamides as Axl kinase inhibitors utilizing a Mer mutant surrogate. Bioorg. Med. Chem. Lett., 27, 2017