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PDB: 1 results

5KR7
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BU of 5kr7 by Molmil
KDM4C bound to pyrazolo-pyrimidine scaffold
Descriptor: 6-ethyl-2,5-dimethyl-7-oxidanylidene-4~{H}-pyrazolo[1,5-a]pyrimidine-3-carbonitrile, CHLORIDE ION, FE (II) ION, ...
Authors:Bellon, S.F, Poy, F, Setser, J.W.
Deposit date:2016-07-07
Release date:2016-08-17
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Identification of potent, selective KDM5 inhibitors.
Bioorg.Med.Chem.Lett., 26, 2016

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