PDB Search results for query - Protein Data Bank Japan

PDB: 2 results

Crystal structure of human Pim-1 kinase in complex with a thiazolamine-indazole inhibitor.
Descriptor:	5-[3-(quinolin-3-yl)-2H-indazol-5-yl]-1,3-thiazol-2-amine, GLYCEROL, Serine/threonine-protein kinase pim-1
Authors:	Mohr, C.
Deposit date:	2014-10-28
Release date:	2015-02-11
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (2.3 Å)
Cite:	Discovery of 5-(1H-indol-5-yl)-1,3,4-thiadiazol-2-amines as potent PIM inhibitors. Bioorg.Med.Chem.Lett., 25, 2015

Crystal structure of human Pim-1 kinase in complex with a thiadiazolamine-indole inhibitor.
Descriptor:	6-[5-(5-amino-1,3,4-thiadiazol-2-yl)-1H-indol-3-yl]-N-cyclopentylpyridin-2-amine, GLYCEROL, Serine/threonine-protein kinase pim-1
Authors:	Mohr, C.
Deposit date:	2014-10-29
Release date:	2015-02-11
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (2.3 Å)
Cite:	Discovery of 5-(1H-indol-5-yl)-1,3,4-thiadiazol-2-amines as potent PIM inhibitors. Bioorg.Med.Chem.Lett., 25, 2015