English
日本語
简体中文
繁體中文
한국어
✖
Menu
RCSB PDB
PDBe
BMRB
Adv. Search
Search help
PDB: 2 results
1RWX
Crystal structure of human caspase-1 in complex with 4-oxo-3-{6-[4-(quinoxalin-2-yloxy)-benzoylamino]-2-thiophen-2-yl-hexanoylamino}-butyric acid
Descriptor:
4-OXO-3-{6-[4-(QUINOXALIN-2-YLOXY)-BENZOYLAMINO]-2-THIOPHEN-2-YL-HEXANOYLAMINO}-BUTYRIC ACID, Interleukin-1 beta convertase
Authors:
Romanowski, M.J
,
Fahr, B.T
,
O'Brien, T.
Deposit date:
2003-12-17
Release date:
2004-12-28
Last modified:
2023-08-23
Method:
X-RAY DIFFRACTION (1.85 Å)
Cite:
Tethering identifies fragment that yields potent inhibitors of human caspase-1.
Bioorg.Med.Chem.Lett., 16, 2006
1RWW
Crystal structure of human caspase-1 in complex with 4-oxo-3-[(6-{[4-(quinoxalin-2-ylamino)-benzoylamino]-methyl}-pyridine-3-carbonyl)-amino]-butyric acid
Descriptor:
4-OXO-3-[(6-{[4-(QUINOXALIN-2-YLAMINO)-BENZOYLAMINO]-METHYL}-PYRIDINE-3-CARBONYL)-AMINO]-BUTYRIC ACID, Interleukin-1 beta convertase
Authors:
Romanowski, M.J
,
Fahr, B.T
,
O'Brien, T.
Deposit date:
2003-12-17
Release date:
2004-12-28
Last modified:
2023-08-23
Method:
X-RAY DIFFRACTION (2.8 Å)
Cite:
Tethering identifies fragment that yields potent inhibitors of human caspase-1.
Bioorg.Med.Chem.Lett., 16, 2006
Home
Top Page
Statistics
Help
FAQ
Contact Us
Cite Us / Terms and Conditions
Links
Settings
Data deposition (OneDep)
Help
Deposition to PDB, EMDB or BMRB
Download
Download PDB archive / snapshot archive
Standard format
PDBx/mmCIF Resources
Format Conversion
PDBx/mmCIF editor
Quick links
Help
non-PDB format compatible
Group Depositions
Chemical Component entries
Latest entries
Search services
Help
Search PDB (PDBj Mine)
Search PDBj RDB
Chemie search
Search BMRB
Sequence-Navigator
DASH
EM Navigator
Omokage search
SeSAW
wwPDB/RDF
RDF Portal
Status search
Molecular Viewers
Help
jV: Graphic Viewer
Molmil: WebGL Mol. Viewer
Services & Softwares
Help
Yorodumi
ASH
MAFFTash
NMRToolBox
gmfit
CRNPRED
Spanner
SFAS
HOMCOS
Derived databases
Help
eF-site
eF-seek
eF-surf
ProMode Elastic
hGTOP
Educational service
Help
eProtS
Molecule of the Month
Previous workshop
Games
Papermodels
About PDBj
Help
Publications
Newsletters / Public Relations Resources
PDBj Members
PDBj Advisory Committee
Privacy Policy
222415
PDB entries from 2024-07-10