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PDB: 1 results

4XY2
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BU of 4xy2 by Molmil
Crystal structure of PDE10A in complex with ASP9436
Descriptor: 1-methyl-5-(1-methyl-3-{[4-(1-methyl-1H-benzimidazol-4-yl)phenoxy]methyl}-1H-pyrazol-4-yl)pyridin-2(1H)-one, MAGNESIUM ION, ZINC ION, ...
Authors:Amano, Y, Honbou, K.
Deposit date:2015-02-02
Release date:2015-06-17
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (2.03 Å)
Cite:Addressing phototoxicity observed in a novel series of biaryl derivatives: Discovery of potent, selective and orally active phosphodiesterase 10A inhibitor ASP9436
Bioorg.Med.Chem., 23, 2015

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