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PDB: 2 results

8VA6
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BU of 8va6 by Molmil
Menin in complex with Ziftomenib (KO-539)
Descriptor: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, DIMETHYL SULFOXIDE, ...
Authors:Clegg, B.D, Linhares, B.M, Cierpicki, T, Grembecka, J.
Deposit date:2023-12-11
Release date:2024-11-20
Last modified:2025-06-04
Method:X-RAY DIFFRACTION (1.57 Å)
Cite:Ziftomenib in relapsed or refractory acute myeloid leukaemia (KOMET-001): a multicentre, open-label, multi-cohort, phase 1 trial.
Lancet Oncol, 25, 2024
8VA5
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BU of 8va5 by Molmil
Menin mutant - T349M in complex with Ziftomenib (KO-539)
Descriptor: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, DIMETHYL SULFOXIDE, ...
Authors:Clegg, B.D, Cierpicki, T, Grembecka, J.
Deposit date:2023-12-11
Release date:2024-11-20
Last modified:2025-06-04
Method:X-RAY DIFFRACTION (1.3 Å)
Cite:Ziftomenib in relapsed or refractory acute myeloid leukaemia (KOMET-001): a multicentre, open-label, multi-cohort, phase 1 trial.
Lancet Oncol, 25, 2024

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PDB entries from 2025-07-30

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