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PDB: 1 results
3R8D
Activation of the Human Nuclear Xenobiotic Receptor PXR by the Reverse Transcriptase-Targeted Anti-HIV Drug PNU-142721
Descriptor:
6-CHLORO-2-(1-FURO[2,3-C]PYRIDIN-5-YL-ETHYLSULFANYL)-PYRIMIDIN-4-YLAMINE, Nuclear receptor subfamily 1 group I member 2
Authors:
Cheng, Y
,
Redinbo, M.R.
Deposit date:
2011-03-23
Release date:
2011-08-17
Last modified:
2024-02-21
Method:
X-RAY DIFFRACTION (2.8 Å)
Cite:
Activation of the human nuclear xenobiotic receptor PXR by the reverse transcriptase-targeted anti-HIV drug PNU-142721.
Protein Sci., 20, 2011
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PDB entries from 2024-07-24