9FM5
 
 | PvSub1 Catalytic Domain in Complex with Peptidomimetic Inhibitor (AL-97) | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 5,6-DIHYDRO-BENZO[H]CINNOLIN-3-YLAMINE, CALCIUM ION, ... | Authors: | Batista, F.A, Martinez, M, Bouillon, A, Mechaly, A, Alzari, P.M, Haouz, A, Barale, J.C. | Deposit date: | 2024-06-05 | Release date: | 2025-02-05 | Last modified: | 2025-04-30 | Method: | X-RAY DIFFRACTION (1.597 Å) | Cite: | Towards Improved Peptidic alpha-Ketoamide Inhibitors of the Plasmodial Subtilisin-Like SUB1: Exploration of N-Terminal Extensions and Cyclic Constraints. Chemmedchem, 20, 2025
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