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7LH8
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CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH INHIBITOR JJ-II-131
Descriptor: (5R)-1-ethyl-5-(4-methylphenyl)-7-({1-[(4-nitrophenyl)methyl]piperidin-4-yl}methyl)-5,7,8,9-tetrahydro-1H-pyrrolo[3',4':5,6]pyrido[2,3-d]pyrimidine-2,4,6(3H)-trione, 1,2-ETHANEDIOL, Bromodomain-containing protein 4, ...
Authors:Schonbrunn, E, Chan, A.
Deposit date:2021-01-21
Release date:2022-07-06
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (1.75 Å)
Cite:Dihydropyridine Lactam Analogs Targeting BET Bromodomains.
Chemmedchem, 17, 2022

221051

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