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PDB: 1 results
5NGB
X-Ray Diffraction Crystal Structure of the murine PI3K p110delta in complex with a pan inhibitor
Descriptor:
3-[[4-(2-morpholin-4-yl-4-oxidanylidene-3~{H}-quinolin-8-yl)-1,2,3-triazol-1-yl]methyl]benzoic acid, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Authors:
Berndt, A
,
Williams, R.L.
Deposit date:
2017-03-17
Release date:
2017-09-13
Last modified:
2024-01-17
Method:
X-RAY DIFFRACTION (2.9 Å)
Cite:
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs.
ChemMedChem, 12, 2017
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PDB entries from 2024-07-10