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PDB: 2 results

5LXP
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BU of 5lxp by Molmil
Human PARP14 (ARTD8), catalytic fragment in complex with inhibitor H5
Descriptor: Poly [ADP-ribose] polymerase 14, ~{N}'-(3-aminocarbonylphenyl)-~{N}-[[1-[(2~{R})-2-phenylpropyl]-1,2,3-triazol-4-yl]methyl]pentanediamide
Authors:Karlberg, T, Thorsell, A.G, Schuler, H.
Deposit date:2016-09-22
Release date:2016-12-21
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.07 Å)
Cite:Small Molecule Microarray Based Discovery of PARP14 Inhibitors.
Angew. Chem. Int. Ed. Engl., 56, 2017
5LYH
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BU of 5lyh by Molmil
Human PARP14 (ARTD8), catalytic fragment in complex with inhibitor H10
Descriptor: 3-[2-[4-[2-[[4-[(3-aminocarbonylphenyl)amino]-4-oxidanylidene-butanoyl]amino]ethyl]-1,2,3-triazol-1-yl]ethylsulfamoyl]benzoic acid, Poly [ADP-ribose] polymerase 14
Authors:Karlberg, T, Thorsell, A.G, Schuler, H.
Deposit date:2016-09-28
Release date:2016-12-21
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.17 Å)
Cite:Small Molecule Microarray Based Discovery of PARP14 Inhibitors.
Angew. Chem. Int. Ed. Engl., 56, 2017

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