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Crystal structure of PqsR (MvfR) ligand-binding domain in complex with 3-PYRIDIN-4-YL-2,4-DIHYDRO-INDENO[1,2-.C.]PYRAZOLE
Descriptor:	Transcriptional regulator MvfR, ~{N}-[[2-(3-chloranyl-4-propan-2-yloxy-phenyl)pyrimidin-5-yl]methyl]-2-(trifluoromethyl)pyridin-4-amine
Authors:	Schmelz, S, Blankenfeldt, W.
Deposit date:	2021-07-13
Release date:	2022-07-27
Last modified:	2024-01-31
Method:	X-RAY DIFFRACTION (2.74 Å)
Cite:	Towards Translation of PqsR Inverse Agonists: From In Vitro Efficacy Optimization to In Vivo Proof-of-Principle. Adv Sci, 10, 2023