9BK2
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![BU of 9bk2 by Molmil](/molmil-images/mine/9bk2) | Crystal structure of Lactate dehydrogenase in complex with 4-((4-(1-methyl-1H-imidazole-2-carbonyl)phenyl)amino)-4-oxo-2-(4-(trifluoromethyl)phenyl)butanoic acid (S-enantiomer, monoclinic P form) | Descriptor: | (2S)-4-[4-(1-methyl-1H-imidazole-2-carbonyl)anilino]-4-oxo-2-[4-(trifluoromethyl)phenyl]butanoic acid, DIMETHYL SULFOXIDE, L-lactate dehydrogenase A chain, ... | Authors: | Lovell, S, Cooper, A, Battaile, K.P, Sharma, H, Seattle Structural Genomics Center for Infectious Disease (SSGCID) | Deposit date: | 2024-04-26 | Release date: | 2024-07-10 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Synthesis and biological characterization of an orally bioavailable lactate dehydrogenase-A inhibitor against pancreatic cancer. Eur.J.Med.Chem., 275, 2024
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9B35
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![BU of 9b35 by Molmil](/molmil-images/mine/9b35) | Ligand-binding and transmembrane domains of kainate receptor GluK2 in the open state, a complex with agonist glutamate and positive allosteric modulator BPAM344 | Descriptor: | GLUTAMIC ACID, Glutamate receptor ionotropic, kainate 2 | Authors: | Nadezhdin, K.D, Gangwar, S.P, Sobolevsky, A.I. | Deposit date: | 2024-03-18 | Release date: | 2024-05-22 | Last modified: | 2024-06-26 | Method: | ELECTRON MICROSCOPY (3.4 Å) | Cite: | Kainate receptor channel opening and gating mechanism. Nature, 630, 2024
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8UP3
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![BU of 8up3 by Molmil](/molmil-images/mine/8up3) | Structure of atypical asparaginase from Rhodospirillum rubrum (mutant Y21F) | Descriptor: | 1,2-ETHANEDIOL, ASPARTIC ACID, Asparaginase, ... | Authors: | Lubkowski, J, Wlodawer, A, Zhang, D. | Deposit date: | 2023-10-20 | Release date: | 2024-04-03 | Method: | X-RAY DIFFRACTION (1.76 Å) | Cite: | RrA, an enzyme from Rhodospirillum rubrum, is a prototype of a new family of short-chain L-asparaginases. Protein Sci., 33, 2024
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9AXH
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![BU of 9axh by Molmil](/molmil-images/mine/9axh) | Crystal structure of KSR1/MEK1 complex heterotetramer with NST-628 | Descriptor: | 1,2-ETHANEDIOL, CHLORIDE ION, Dual specificity mitogen-activated protein kinase kinase 1, ... | Authors: | Quade, B, Huang, X. | Deposit date: | 2024-03-06 | Release date: | 2024-04-17 | Last modified: | 2024-07-10 | Method: | X-RAY DIFFRACTION (2.81 Å) | Cite: | The Pan-RAF-MEK Nondegrading Molecular Glue NST-628 Is a Potent and Brain-Penetrant Inhibitor of the RAS-MAPK Pathway with Activity across Diverse RAS- and RAF-Driven Cancers. Cancer Discov, 14, 2024
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9BK3
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![BU of 9bk3 by Molmil](/molmil-images/mine/9bk3) | Crystal structure of Lactate dehydrogenase in complex with 4-((4-(1-methyl-1H-imidazole-2-carbonyl)phenyl)amino)-4-oxo-2-(4-(trifluoromethyl)phenyl)butanoic acid (R-enantiomer, orthorhombic P form) | Descriptor: | (2R)-4-[4-(1-methyl-1H-imidazole-2-carbonyl)anilino]-4-oxo-2-[4-(trifluoromethyl)phenyl]butanoic acid, CHLORIDE ION, L-lactate dehydrogenase A chain, ... | Authors: | Lovell, S, Cooper, A, Battaile, K.P, Sharma, H. | Deposit date: | 2024-04-26 | Release date: | 2024-07-10 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | Synthesis and biological characterization of an orally bioavailable lactate dehydrogenase-A inhibitor against pancreatic cancer. Eur.J.Med.Chem., 275, 2024
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8UPC
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![BU of 8upc by Molmil](/molmil-images/mine/8upc) | Structure of atypical asparaginase from Rhodospirillum rubrum (mutant K158M) | Descriptor: | Asparaginase, CHLORIDE ION, GLYCEROL | Authors: | Lubkowski, J, Wlodawer, A, Zhang, D. | Deposit date: | 2023-10-22 | Release date: | 2024-04-03 | Method: | X-RAY DIFFRACTION (1.2 Å) | Cite: | RrA, an enzyme from Rhodospirillum rubrum, is a prototype of a new family of short-chain L-asparaginases. Protein Sci., 33, 2024
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9B5V
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8WT1
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![BU of 8wt1 by Molmil](/molmil-images/mine/8wt1) | Crystal structure of S9 carboxypeptidase from Geobacillus sterothermophilus | Descriptor: | ALANINE, CITRATE ANION, GLYCEROL, ... | Authors: | Chandravanshi, K, Kumar, A, Sen, C, Singh, R, Bhange, G.B, Makde, R.D. | Deposit date: | 2023-10-17 | Release date: | 2024-03-13 | Last modified: | 2024-04-10 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Crystal structure and solution scattering of Geobacillus stearothermophilus S9 peptidase reveal structural adaptations for carboxypeptidase activity. Febs Lett., 598, 2024
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9B5T
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![BU of 9b5t by Molmil](/molmil-images/mine/9b5t) | |
9ASL
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![BU of 9asl by Molmil](/molmil-images/mine/9asl) | |
9B56
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![BU of 9b56 by Molmil](/molmil-images/mine/9b56) | |
8UOO
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![BU of 8uoo by Molmil](/molmil-images/mine/8uoo) | Structure of atypical asparaginase from Rhodospirillum rubrum | Descriptor: | Asparaginase, CHLORIDE ION, GLYCEROL | Authors: | Lubkowski, J, Wlodawer, A, Zhang, D. | Deposit date: | 2023-10-20 | Release date: | 2024-04-03 | Method: | X-RAY DIFFRACTION (1.65 Å) | Cite: | RrA, an enzyme from Rhodospirillum rubrum, is a prototype of a new family of short-chain L-asparaginases. Protein Sci., 33, 2024
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8UP7
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![BU of 8up7 by Molmil](/molmil-images/mine/8up7) | Structure of atypical asparaginase from Rhodospirillum rubrum (mutant K19A) | Descriptor: | Asparaginase, CHLORIDE ION | Authors: | Lubkowski, J, Wlodawer, A, Zhang, D. | Deposit date: | 2023-10-21 | Release date: | 2024-04-03 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | RrA, an enzyme from Rhodospirillum rubrum, is a prototype of a new family of short-chain L-asparaginases. Protein Sci., 33, 2024
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8UP9
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![BU of 8up9 by Molmil](/molmil-images/mine/8up9) | Structure of atypical asparaginase from Rhodospirillum rubrum (mutant K19Q) | Descriptor: | 1,2-ETHANEDIOL, Asparaginase, CHLORIDE ION, ... | Authors: | Lubkowski, J, Wlodawer, A, Zhang, D. | Deposit date: | 2023-10-21 | Release date: | 2024-04-03 | Method: | X-RAY DIFFRACTION (1.47 Å) | Cite: | RrA, an enzyme from Rhodospirillum rubrum, is a prototype of a new family of short-chain L-asparaginases. Protein Sci., 33, 2024
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3VET
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![BU of 3vet by Molmil](/molmil-images/mine/3vet) | Crystal structure of the O-carbamoyltransferase TobZ in complex with Tobramycin, carbamoyl phosphate and ADP | Descriptor: | 1,2-ETHANEDIOL, ADENOSINE-5'-DIPHOSPHATE, FE (II) ION, ... | Authors: | Parthier, C, Stubbs, M.T, Goerlich, S, Jaenecke, F. | Deposit date: | 2012-01-09 | Release date: | 2012-01-25 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | The O-Carbamoyltransferase TobZ Catalyzes an Ancient Enzymatic Reaction. Angew.Chem.Int.Ed.Engl., 51, 2012
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8UOR
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![BU of 8uor by Molmil](/molmil-images/mine/8uor) | Structure of atypical asparaginase from Rhodospirillum rubrum (mutant K19E) | Descriptor: | 1,2-ETHANEDIOL, Asparaginase, CHLORIDE ION | Authors: | Lubkowski, J, Wlodawer, A, Zhang, D. | Deposit date: | 2023-10-20 | Release date: | 2024-04-03 | Method: | X-RAY DIFFRACTION (1.45 Å) | Cite: | RrA, an enzyme from Rhodospirillum rubrum, is a prototype of a new family of short-chain L-asparaginases. Protein Sci., 33, 2024
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9B58
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![BU of 9b58 by Molmil](/molmil-images/mine/9b58) | |
8ZKV
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![BU of 8zkv by Molmil](/molmil-images/mine/8zkv) | |
9B5N
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![BU of 9b5n by Molmil](/molmil-images/mine/9b5n) | |
1A1A
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![BU of 1a1a by Molmil](/molmil-images/mine/1a1a) | |
9B5R
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9B5P
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9B5S
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![BU of 9b5s by Molmil](/molmil-images/mine/9b5s) | |
8UOU
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![BU of 8uou by Molmil](/molmil-images/mine/8uou) | Structure of atypical asparaginase from Rhodospirillum rubrum in complex with L-Asp | Descriptor: | ASPARTIC ACID, Asparaginase, CHLORIDE ION | Authors: | Lubkowski, J, Wlodawer, A, Zhang, D. | Deposit date: | 2023-10-20 | Release date: | 2024-04-03 | Method: | X-RAY DIFFRACTION (1.35 Å) | Cite: | RrA, an enzyme from Rhodospirillum rubrum, is a prototype of a new family of short-chain L-asparaginases. Protein Sci., 33, 2024
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9B5X
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![BU of 9b5x by Molmil](/molmil-images/mine/9b5x) | |