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PDB: 1 results

3TWJ
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Rho-associated protein kinase 1 (ROCK 1) IN COMPLEX WITH RKI1447
Descriptor: 1,2-ETHANEDIOL, 1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea, Rho-associated protein kinase 1
Authors:Martin, M.P, Zhu, J.-Y, Schonbrunn, E.
Deposit date:2011-09-21
Release date:2012-08-22
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:RKI-1447 Is a Potent Inhibitor of the Rho-Associated ROCK Kinases with Anti-Invasive and Antitumor Activities in Breast Cancer.
Cancer Res., 72, 2012

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數據於2024-07-24公開中

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