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PDB: 1 results

6GVA
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BU of 6gva by Molmil
CDK2/cyclin A2 in complex with pyrazolo[4,3-d]pyrimidine inhibitor LGR4455
Descriptor: 1,2-ETHANEDIOL, 5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{N}-[(4-pyridin-2-ylphenyl)methyl]-2~{H}-pyrazolo[4,3-d]pyrimidin-7-amine, BROMIDE ION, ...
Authors:Skerlova, J, Rezacova, P.
Deposit date:2018-06-20
Release date:2019-05-01
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:3,5,7-Substituted Pyrazolo[4,3- d]pyrimidine Inhibitors of Cyclin-Dependent Kinases and Their Evaluation in Lymphoma Models.
J.Med.Chem., 62, 2019

222415

數據於2024-07-10公開中

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