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PDB: 2 results
6PL2
TRK-A IN COMPLEX WITH LIGAND 1a
Descriptor:
High affinity nerve growth factor receptor, N-(3-tert-butyl-1-phenyl-1H-pyrazol-5-yl)-2-{[1-(4-hydroxyphenyl)-1H-tetrazol-5-yl]sulfanyl}acetamide
Authors:
Subramanian, G.
Deposit date:
2019-06-30
Release date:
2019-09-04
Last modified:
2019-09-25
Method:
X-RAY DIFFRACTION (2.59 Å)
Cite:
Type 2 inhibitor leads of human tropomyosin receptor kinase (hTrkA).
Bioorg.Med.Chem.Lett., 29, 2019
6PL3
TRK-A IN COMPLEX WITH LIGAND 2a
Descriptor:
2-[(3-tert-butyl-1-phenyl-1H-pyrazol-5-yl)amino]-2-oxoethyl 4-(1H-tetrazol-1-yl)benzoate, High affinity nerve growth factor receptor
Authors:
Subramanian, G.
Deposit date:
2019-06-30
Release date:
2019-09-04
Last modified:
2024-03-13
Method:
X-RAY DIFFRACTION (3 Å)
Cite:
Type 2 inhibitor leads of human tropomyosin receptor kinase (hTrkA).
Bioorg.Med.Chem.Lett., 29, 2019
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223532
數據於2024-08-07公開中