5KQF
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![BU of 5kqf by Molmil](/molmil-images/mine/5kqf) | (4~{S},6~{S})-4-[2,4-bis(fluoranyl)phenyl]-4-methyl-6-pyrimidin-5-yl-5,6-dihydro-1,3-thiazin-2-amine (compound 12) bound to BACE1 | Descriptor: | (4~{S},6~{S})-4-[2,4-bis(fluoranyl)phenyl]-4-methyl-6-pyrimidin-5-yl-5,6-dihydro-1,3-thiazin-2-amine, Beta-secretase 1 | Authors: | Lewis, H.A, Wu, Y.J, Rajamani, R, Thompson, L.A. | Deposit date: | 2016-07-06 | Release date: | 2016-09-07 | Last modified: | 2016-10-05 | Method: | X-RAY DIFFRACTION (1.98 Å) | Cite: | Discovery of S3-Truncated, C-6 Heteroaryl Substituted Aminothiazine beta-Site APP Cleaving Enzyme-1 (BACE1) Inhibitors. J.Med.Chem., 59, 2016
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5KR8
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![BU of 5kr8 by Molmil](/molmil-images/mine/5kr8) | (4~{S},6~{S})-4-[2,4-bis(fluoranyl)phenyl]-6-(3,5-dimethyl-1,2-oxazol-4-yl)-4-methyl-5,6-dihydro-1,3-thiazin-2-amine (compound 5) bound to BACE1 | Descriptor: | (4~{S},6~{S})-4-[2,4-bis(fluoranyl)phenyl]-6-(3,5-dimethyl-1,2-oxazol-4-yl)-4-methyl-5,6-dihydro-1,3-thiazin-2-amine, Beta-secretase 1, IODIDE ION | Authors: | Lewis, H.A, Wu, Y.J, Rajamani, R, Thompson, L.A. | Deposit date: | 2016-07-07 | Release date: | 2016-09-07 | Last modified: | 2016-10-05 | Method: | X-RAY DIFFRACTION (2.118 Å) | Cite: | Discovery of S3-Truncated, C-6 Heteroaryl Substituted Aminothiazine beta-Site APP Cleaving Enzyme-1 (BACE1) Inhibitors. J.Med.Chem., 59, 2016
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5JOD
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![BU of 5jod by Molmil](/molmil-images/mine/5jod) | Structure of proplasmepsin IV from Plasmodium falciparum | Descriptor: | GLYCEROL, Proplasmepsin IV | Authors: | Recacha, R, Akopjana, I, Tars, K, Jaudzems, K. | Deposit date: | 2016-05-02 | Release date: | 2016-08-17 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (1.528 Å) | Cite: | Crystal structure of Plasmodium falciparum proplasmepsin IV: the plasticity of proplasmepsins. Acta Crystallogr.,Sect.F, 72, 2016
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5P7D
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![BU of 5p7d by Molmil](/molmil-images/mine/5p7d) | |
5P7T
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![BU of 5p7t by Molmil](/molmil-images/mine/5p7t) | |
5P86
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![BU of 5p86 by Molmil](/molmil-images/mine/5p86) | |
5P8L
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![BU of 5p8l by Molmil](/molmil-images/mine/5p8l) | |
5OZ6
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![BU of 5oz6 by Molmil](/molmil-images/mine/5oz6) | |
5OZH
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![BU of 5ozh by Molmil](/molmil-images/mine/5ozh) | |
5OZB
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![BU of 5ozb by Molmil](/molmil-images/mine/5ozb) | |
5OZP
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![BU of 5ozp by Molmil](/molmil-images/mine/5ozp) | |
5P03
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![BU of 5p03 by Molmil](/molmil-images/mine/5p03) | |
5P0I
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![BU of 5p0i by Molmil](/molmil-images/mine/5p0i) | |
5P0U
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![BU of 5p0u by Molmil](/molmil-images/mine/5p0u) | |
5P19
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![BU of 5p19 by Molmil](/molmil-images/mine/5p19) | |
5P1P
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![BU of 5p1p by Molmil](/molmil-images/mine/5p1p) | |
5P23
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![BU of 5p23 by Molmil](/molmil-images/mine/5p23) | |
5P2F
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![BU of 5p2f by Molmil](/molmil-images/mine/5p2f) | |
5P2T
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![BU of 5p2t by Molmil](/molmil-images/mine/5p2t) | |
5P35
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![BU of 5p35 by Molmil](/molmil-images/mine/5p35) | |
5P3L
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![BU of 5p3l by Molmil](/molmil-images/mine/5p3l) | |
5P40
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![BU of 5p40 by Molmil](/molmil-images/mine/5p40) | |
5P4I
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![BU of 5p4i by Molmil](/molmil-images/mine/5p4i) | |
5P51
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![BU of 5p51 by Molmil](/molmil-images/mine/5p51) | |
5P5H
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![BU of 5p5h by Molmil](/molmil-images/mine/5p5h) | |