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4WNK
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Crystal Structure of Bovine G Protein Coupled-Receptor Kinase 5 in Complex with CCG215022
Descriptor: (4S)-4-{4-fluoro-3-[(pyridin-2-ylmethyl)carbamoyl]phenyl}-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide, G protein-coupled receptor kinase 5, SULFATE ION
Authors:Homan, K.T, Tesmer, J.J.G.
Deposit date:2014-10-13
Release date:2015-06-10
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.42 Å)
Cite:Crystal Structure of G Protein-coupled Receptor Kinase 5 in Complex with a Rationally Designed Inhibitor.
J.Biol.Chem., 290, 2015

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数据于2024-07-10公开中

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