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PDB: 3 results

6XER
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BU of 6xer by Molmil
Tubulin-RB3_SLD in complex with colchicine
Descriptor: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
Authors:White, S.W, Yun, M.
Deposit date:2020-06-13
Release date:2021-08-25
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Design, Synthesis, and Biological Evaluation of Stable Colchicine-Binding Site Tubulin Inhibitors 6-Aryl-2-benzoyl-pyridines as Potential Anticancer Agents.
J.Med.Chem., 64, 2021
6XET
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BU of 6xet by Molmil
Tubulin-RB3_SLD in complex with compound 60c
Descriptor: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
Authors:White, S.W, Yun, M.
Deposit date:2020-06-13
Release date:2021-08-25
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Design, Synthesis, and Biological Evaluation of Stable Colchicine-Binding Site Tubulin Inhibitors 6-Aryl-2-benzoyl-pyridines as Potential Anticancer Agents.
J.Med.Chem., 64, 2021
6XES
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BU of 6xes by Molmil
Tubulin-RB3_SLD in complex with compound 40a
Descriptor: DIMETHYL SULFOXIDE, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
Authors:White, S.W, Yun, M.
Deposit date:2020-06-13
Release date:2021-08-25
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.32 Å)
Cite:Design, Synthesis, and Biological Evaluation of Stable Colchicine-Binding Site Tubulin Inhibitors 6-Aryl-2-benzoyl-pyridines as Potential Anticancer Agents.
J.Med.Chem., 64, 2021

222624

数据于2024-07-17公开中

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