3ESS
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2Q6M
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3KI3
| Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-H | Descriptor: | 2-[(dimethylamino)methyl]-5,6-dihydroimidazo[4,5,1-jk][1,4]benzodiazepin-7(4H)-one, Cholix toxin | Authors: | Jorgensen, R, Edwards, P.R, Merrill, A.R. | Deposit date: | 2009-10-31 | Release date: | 2010-10-27 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.27 Å) | Cite: | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
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3KI2
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3KI0
| Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-D | Descriptor: | 3-(morpholin-4-ylmethyl)-1,5-dihydro-6H-[1,2]diazepino[4,5,6-cd]indol-6-one, CHLORIDE ION, Cholix toxin | Authors: | Jorgensen, R, Edwards, P.R, Merrill, A.R. | Deposit date: | 2009-10-31 | Release date: | 2010-10-27 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.29 Å) | Cite: | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
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3KI7
| Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-I | Descriptor: | 2-{2-[4-(pyrrolidin-1-ylmethyl)phenyl]ethyl}-5,6-dihydroimidazo[4,5,1-jk][1,4]benzodiazepin-7(4H)-one, Cholix toxin | Authors: | Jorgensen, R, Edwards, P.R, Merrill, A.R. | Deposit date: | 2009-10-31 | Release date: | 2010-10-27 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.32 Å) | Cite: | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
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3KI1
| Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-F | Descriptor: | 2-{4-[3-(dimethylamino)propoxy]phenyl}-5,6-dihydroimidazo[4,5,1-jk][1,4]benzodiazepin-7(4H)-one, Cholix toxin | Authors: | Jorgensen, R, Edwards, P.R, Merrill, A.R. | Deposit date: | 2009-10-31 | Release date: | 2010-10-27 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.43 Å) | Cite: | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
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3KI6
| Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-L | Descriptor: | 8-fluoro-2-(3-piperidin-1-ylpropanoyl)-1,3,4,5-tetrahydrobenzo[c][1,6]naphthyridin-6(2H)-one, Cholix toxin | Authors: | Jorgensen, R, Edwards, P.R, Merrill, A.R. | Deposit date: | 2009-10-31 | Release date: | 2010-10-27 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.54 Å) | Cite: | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
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3KI5
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3KI4
| Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-P | Descriptor: | (11bR)-3-oxo-1,2,3,11b-tetrahydrochromeno[4,3,2-de]isoquinoline-10-sulfonic acid, Cholix toxin, GLYCEROL | Authors: | Jorgensen, R, Edwards, P.R, Merrill, A.R. | Deposit date: | 2009-10-31 | Release date: | 2010-10-27 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.65 Å) | Cite: | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
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3NY6
| Catalytic fragment of cholix toxin from vibrio cholerae in complex with inhibitor V30 | Descriptor: | 2-[(5,6-dimethyl-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(2-hydroxyethyl)acetamide, Cholix toxin, GLYCEROL, ... | Authors: | Merrill, A.R, Jorgensen, R. | Deposit date: | 2010-07-14 | Release date: | 2010-12-29 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.68 Å) | Cite: | Newly discovered and characterized antivirulence compounds inhibit bacterial mono-ADP-ribosyltransferase toxins. Antimicrob.Agents Chemother., 55, 2011
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3Q9O
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2Q5T
| Full-length Cholix toxin from Vibrio Cholerae | Descriptor: | 1,2-ETHANEDIOL, CHLORIDE ION, Cholix toxin | Authors: | Jorgensen, R, Fieldhouse, R.J, Merrill, A.R. | Deposit date: | 2007-06-01 | Release date: | 2008-02-12 | Last modified: | 2023-08-30 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Cholix Toxin, a Novel ADP-ribosylating Factor from Vibrio cholerae. J.Biol.Chem., 283, 2008
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