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PDB: 1 results

4KRS
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BU of 4krs by Molmil
Tankyrase-1 complexed with small molecule inhibitor
Descriptor: 4-tert-butyl-N-(5,6-dihydro[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl)benzamide, SULFATE ION, Tankyrase-1, ...
Authors:Stams, T, Kirby, C.
Deposit date:2013-05-17
Release date:2013-08-28
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.29 Å)
Cite:Structure-Efficiency Relationship of [1,2,4]Triazol-3-ylamines as Novel Nicotinamide Isosteres that Inhibit Tankyrases.
J.Med.Chem., 56, 2013

222415

건을2024-07-10부터공개중

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