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8BPY
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X-RAY STRUCTURE OF PDE9A IN COMPLEX WITH Inhibitor 13A
Descriptor: (8~{S})-6-[2-(2,3-dihydroindol-1-yl)-2-oxidanylidene-ethyl]-4-(4-methylphenyl)-2-oxidanylidene-8-propyl-1,5,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile, High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A, MAGNESIUM ION, ...
Authors:Steuber, H.
Deposit date:2022-11-18
Release date:2022-12-28
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (3.3 Å)
Cite:BAY-7081: A Potent, Selective, and Orally Bioavailable Cyanopyridone-Based PDE9A Inhibitor.
J.Med.Chem., 65, 2022

222415

건을2024-07-10부터공개중

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