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PDB: 1 results

5T19
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BU of 5t19 by Molmil
Structure of PTP1B complexed with N-(3'-(1,1-dioxido-4-oxo-1,2,5-thiadiazolidin-2-yl)-4'-methyl-[1,1'-biphenyl]-4-yl)acetamide
Descriptor: 5-[4-methyl-4'-(methylamino)[1,1'-biphenyl]-3-yl]-1lambda~6~,2,5-thiadiazolidine-1,1,3-trione, CHLORIDE ION, MAGNESIUM ION, ...
Authors:Laciak, A.R, Tanner, J.J.
Deposit date:2016-08-18
Release date:2017-04-12
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.1001 Å)
Cite:Covalent Allosteric Inactivation of Protein Tyrosine Phosphatase 1B (PTP1B) by an Inhibitor-Electrophile Conjugate.
Biochemistry, 56, 2017

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건을2024-07-24부터공개중

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