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PDB: 1 results
7LYE
Myotoxin I from Bothrops moojeni co-crystallized with synthetic inhibitor Varespladib (LY315920)
Descriptor:
({3-[amino(oxo)acetyl]-1-benzyl-2-ethyl-1H-indol-4-yl}oxy)acetic acid, 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, Basic phospholipase A2 homolog BomoTx
Authors:
Salvador, G.H.M
,
Borges, R.J
,
Fontes, M.R.M.
Deposit date:
2021-03-06
Release date:
2021-05-19
Last modified:
2023-10-18
Method:
X-RAY DIFFRACTION (1.758 Å)
Cite:
The synthetic varespladib molecule is a multi-functional inhibitor for PLA 2 and PLA 2 -like ophidic toxins.
Biochim Biophys Acta Gen Subj, 1865, 2021
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